SCHEMBL9325713

SCHEMBL9325713

Nc1nc(Sc2ccccc2)nc2nc(-c3ccoc3)nn12

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.46
ADORA2B P29275 5/20 0.46
ADORA2A P29274 10/20 0.40
ADORA1 P30542 6/20 0.40
CSNK1D P48730 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328686 0.88 ADORA3 (0.42) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9325911 0.84 ADORA3 (0.62) ADORA3ADORA2BADORA2AADORA1
SCHEMBL7828518 0.79 ADORA3 (0.73) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9329166 0.78 ADORA3 (0.41) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9328035 0.77 ADORA3 (0.66) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9325959 0.75 ADORA3 (0.48) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9327033 0.75 ADORA3 (0.51) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9328936 0.74 ADORA3 (0.42) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL23840696 0.72 ADORA3 (0.64) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL23291366 0.72 ADORA2A (0.38) ADORA3ADORA2BADORA2AADORA1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed