SCHEMBL9328686

SCHEMBL9328686

Nc1nc(Sc2ccc(F)cc2)nc2nc(-c3ccoc3)nn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.42
ADORA2B P29275 4/20 0.42
CSNK1D P48730 1/20 0.40
USP2 O75604 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADORA1 P30542 6/20 0.36
ADORA2A P29274 6/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9325713 0.88 ADORA3 (0.46) ADORA3ADORA2BCSNK1DADORA1ADORA2A
SCHEMBL9325911 0.82 ADORA3 (0.62) ADORA3ADORA2BLMNANPC1RAB9A
SCHEMBL9329166 0.76 ADORA3 (0.41) ADORA3ADORA2BCSNK1DUSP2ALDH1A1
SCHEMBL23291366 0.70 ADORA2A (0.38) ADORA3ADORA2BCSNK1DADORA1ADORA2A
SCHEMBL9328035 0.68 ADORA3 (0.66) ADORA3ADORA2BCSNK1DADORA1ADORA2A
SCHEMBL7828518 0.68 ADORA3 (0.73) ADORA3ADORA2BADORA1ADORA2A
SCHEMBL9327228 0.66 ADORA2A (0.67) ADORA3ADORA2BCSNK1DUSP2ALDH1A1
SCHEMBL23963281 0.65 ADORA3 (0.56) ADORA3ADORA2BCSNK1DALDH1A1LMNA
SCHEMBL9325959 0.64 ADORA3 (0.48) ADORA3ADORA2BADORA1ADORA2A
SCHEMBL9327033 0.64 ADORA3 (0.51) ADORA3ADORA2BADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed