SCHEMBL933488

SCHEMBL933488

CC(C)(C)OC(=O)NC1=NCC2COCC[C@]2(c2cccc(N)c2)S1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
AAK1 Q2M2I8 1/20 0.32
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL933050 0.90 HCRTR1 (0.37) HCRTR1HCRTR2AAK1BRD4CREBBP
SCHEMBL932334 0.90 HCRTR1 (0.37) HCRTR1HCRTR2AAK1BRD4CREBBP
SCHEMBL933387 0.86 USP2 (0.34)
SCHEMBL932583 0.82 BACE1 (0.44)
SCHEMBL932766 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1
SCHEMBL6874988 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1
SCHEMBL8028509 0.77 HCRTR1 (0.38) HCRTR1HCRTR2AAK1
SCHEMBL2620087 0.77 HCRTR1 (0.38) HCRTR1HCRTR2AAK1
SCHEMBL932781 0.77 BACE1 (0.32) AAK1
SCHEMBL933505 0.73 CYP1A2 (0.36) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed