SCHEMBL9334455

SCHEMBL9334455

O=C(c1cccc(CN2c3ccccc3Oc3ccccc32)c1)c1c[nH]c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBX7 O95931 1/20 0.47
CDYL2 Q8N8U2 1/20 0.47
CDYL Q9Y232 1/20 0.47
PIM1 P11309 1/20 0.47
GPR84 Q9NQS5 1/20 0.47
RGS12 O14924 1/20 0.44
TP53 P04637 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
MAPK14 Q16539 1/20 0.42
KMT2A Q03164 1/20 0.42
GABRP O00591 3/20 0.41
GABRD O14764 3/20 0.41
GABRA1 P14867 3/20 0.41
GABRB1 P18505 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9337520 0.86 GPR84 (0.49) PIM1GPR84TP53SMN1; SMN2NPSR1
SCHEMBL8793290 0.86 ALDH1A1 (0.47) CBX7CDYL2CDYLPIM1GPR84
SCHEMBL9334005 0.77 KMT2A (0.59) ALDH1A1MAPTHTTKMT2AHDAC3
SCHEMBL1367473 0.74 HDAC6 (0.53) HDAC3HDAC6
SCHEMBL9334431 0.74 SRD5A1 (0.57) KMT2A
SCHEMBL9334424 0.73 TRPA1 (0.55) SMN1; SMN2MAPTHDAC3HDAC6RAB9A
SCHEMBL21366213 0.73 TP53 (0.55) PIM1GPR84TP53SMN1; SMN2NPSR1
SCHEMBL22634965 0.72 GPR84 (0.65) PIM1GPR84TP53SMN1; SMN2NPSR1
SCHEMBL29988308 0.71 GPR84 (0.79) PIM1GPR84TP53SMN1; SMN2NPSR1
SCHEMBL3279652 0.71 GPR84 (0.79) PIM1GPR84TP53SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5312829-A Testosterone 5alpha-reductase inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-05-17 US disclosed
US-5212320-A Enzyme inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-18 US disclosed
EP-0458207-A2 Indole derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-11-27 EP disclosed