SCHEMBL9338202

SCHEMBL9338202

CNCCC(CCC1(c2cc(OC)cc(OC)c2)OCCO1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.38
SLC6A2 P23975 5/20 0.38
CYP2D6 P10635 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NOS2 P35228 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PMP22 Q01453 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ALPL P05186 1/20 0.36
MAPT P10636 1/20 0.36
ALOX12 P18054 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339653 0.86 HTR2A (0.45) SLC6A4SLC6A2CYP2D6MEN1KMT2A
SCHEMBL9341939 0.80 SLC6A4 (0.45) SLC6A4SLC6A2CYP2D6NOS2CYP3A4
SCHEMBL9342579 0.78 ALDH1A1 (0.33) SLC6A4SLC6A2CYP2D6MEN1KMT2A
SCHEMBL9339474 0.77 TP53 (0.38) SLC6A4SLC6A2CYP2D6MEN1KMT2A
Dimethylamine SCHEMBL9337974 0.75 ALDH1A1 (0.40) CYP2D6MEN1KMT2ACYP1A2CYP3A4
SCHEMBL9338360 0.74 SLC6A4 (0.36) SLC6A4SLC6A2CYP2D6MEN1KMT2A
Dimethylamine SCHEMBL9337624 0.72 TSHR (0.40) CYP2D6TSHRHTR2AHRH1ALDH1A1
SCHEMBL9338197 0.71 ICMT (0.34) LMNAALOX12ADRA1AADRA1B
SCHEMBL9342414 0.69 TSHR (0.32) TSHRLMNA
Dimethylamine SCHEMBL9341629 0.67 SLC6A4 (0.46) SLC6A4SLC6A2CYP2D6CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450995-B1 New propanamines, their pharmacological properties and their therapeutical applications, notably as anti-diarrhoea agents JOUVEINAL SA (FR) 1994-06-08 EP disclosed
US-5236947-A Side effect reduction JOUVEINAL S.A. (FR) 1993-08-17 US disclosed
US-5143938-A PROPANAMINES, THEIR PHARMACOLOGICAL PROPERTIES AND THEIR APPLICATION FOR THERAPEUTIC IN PARTICULAR ANTIDIARRHEAL, PURPOSES JOUVEINAL S.A. (FR) 1992-09-01 US disclosed