SCHEMBL934005

SCHEMBL934005

CC(Cc1ccc(OC(F)(F)F)cc1)C(N)=O

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.60
ACACB O00763 1/20 0.53
PTPN1 P18031 1/20 0.48
EPHX2 P34913 5/20 0.46
PPARG P37231 2/20 0.46
PPARA Q07869 2/20 0.46
SCN10A Q9Y5Y9 1/20 0.45
GRIN2B Q13224 1/20 0.45
NR1H4 Q96RI1 1/20 0.44
ACE P12821 1/20 0.44
PLA2G10 O15496 1/20 0.43
PLA2G2A P14555 1/20 0.43
PLA2G5 P39877 1/20 0.43
HRH3 Q9Y5N1 2/20 0.43
FPR2 P25090 2/20 0.43
MAPK8 P45983 1/20 0.43
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24915125 0.86 ACACB (0.54) EPHX1ACACBPTPN1EPHX2PPARG
SCHEMBL15569323 0.86 ACACB (0.54) EPHX1ACACBPTPN1EPHX2PPARG
SCHEMBL934550 0.82 EPHX1 (0.56) EPHX1GRIN2BPLA2G10PLA2G2APLA2G5
SCHEMBL933616 0.82 PPARG (0.59) EPHX1ACACBPTPN1EPHX2PPARG
SCHEMBL14032635 0.82 PPARG (0.60) PTPN1PPARGPPARA
SCHEMBL933857 0.80 LDHA (0.61) EPHX1ACACBPPARGPPARA
SCHEMBL934355 0.80 EPHX1 (0.52) EPHX1ACACBPTPN1EPHX2PPARG
SCHEMBL934143 0.79 EPHX1 (0.45) EPHX1EPHX2PPARGPPARA
SCHEMBL15881521 0.79 CTSD (0.44) EPHX1EPHX2PLA2G10PLA2G2APLA2G5
SCHEMBL1416925 0.78 ACACB (0.52) EPHX1ACACBPTPN1EPHX2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN claimed
WO-2011037833-A2 NOVEL N-BENZYLAMIDE SUBSTITUTED DERIVATIVES OF 2-(ACYLAMIDO)ACETIC ACID AND 2-(ACYLAMIDO)PROPIONIC ACIDS: POTENT NEUROLOGICAL AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2011-03-31 WO disclosed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed
CN-1780821-A Heterocyclic kinase inhibitors. ABBOTT LAB (US) 2006-05-31 CN disclosed