SCHEMBL9340200

SCHEMBL9340200

O=c1c(Br)c(C(F)(F)F)ncn1-c1c(Cl)cc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP3A4 P08684 3/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
HIF1A Q16665 1/20 0.44
TXNRD1 Q16881 1/20 0.44
TXNRD3 Q86VQ6 1/20 0.44
TXNRD2 Q9NNW7 1/20 0.44
CYP2C19 P33261 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
POLB P06746 2/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 2/20 0.36
FGFR4 P22455 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340328 0.92 ALDH1A1 (0.43) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723134 0.88 POLB (0.40) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723076 0.88 TDP1 (0.45) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9339495 0.87 GABRA2 (0.40) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL9723126 0.87 TDP1 (0.44) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9339503 0.87 TDP1 (0.44) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723049 0.85 TDP1 (0.42) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723112 0.85 TDP1 (0.42) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723062 0.84 CYP3A4 (0.42) TDP1ALDH1A1CYP3A4HPGDALOX15
SCHEMBL9723034 0.84 TDP1 (0.41) TDP1ALDH1A1CYP3A4HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0338686-B1 Pyrimidinone derivatives ZENECA LTD (GB) 1994-06-22 EP disclosed
US-5149810-A Chemical intermediates for insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-09-22 US disclosed
US-5104878-A Insecticides, miticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-04-14 US disclosed
US-5077297-A Insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-31 US disclosed
EP-0396250-A1 Pyrimidinone derivatives ZENECA LIMITED (GB) 1990-11-07 EP disclosed
EP-0338686-A2 Pyrimidinone derivatives ZENECA LIMITED (GB) 1989-10-25 EP disclosed