SCHEMBL9723134

SCHEMBL9723134

O=c1c(Br)c(C(F)(F)F)ncn1-c1c([N+](=O)[O-])cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
ALDH1A1 P00352 3/20 0.39
TDP1 Q9NUW8 4/20 0.39
CYP3A4 P08684 4/20 0.39
TSHR P16473 2/20 0.39
HPGD P15428 2/20 0.39
ALOX15 P16050 1/20 0.39
HIF1A Q16665 1/20 0.39
TXNRD1 Q16881 1/20 0.39
TXNRD3 Q86VQ6 1/20 0.39
TXNRD2 Q9NNW7 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
KDM4E B2RXH2 1/20 0.36
PLK1 P53350 1/20 0.36
PTPN5 P54829 1/20 0.34
MAPK1 P28482 4/20 0.34
LMNA P02545 3/20 0.34
MAPT P10636 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340328 0.93 ALDH1A1 (0.43) POLBALDH1A1TDP1CYP3A4TSHR
SCHEMBL9340200 0.88 TDP1 (0.44) POLBALDH1A1TDP1CYP3A4TSHR
SCHEMBL9723045 0.83 HCAR1 (0.36) POLB
SCHEMBL9723061 0.81 GABRA2 (0.37)
SCHEMBL9340421 0.79 CYP3A4 (0.52) POLBALDH1A1TDP1CYP3A4TSHR
SCHEMBL9339513 0.79 ALDH1A1 (0.47) POLBALDH1A1TDP1CYP3A4TSHR
SCHEMBL9723051 0.78 POLB (0.42) POLBALDH1A1TDP1CYP3A4TSHR
SCHEMBL9340204 0.76 HCAR1 (0.30)
SCHEMBL9339495 0.75 GABRA2 (0.40)
SCHEMBL9723076 0.75 TDP1 (0.45) POLBALDH1A1TDP1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5104878-A Insecticides, miticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-04-14 US disclosed
EP-0396250-A1 Pyrimidinone derivatives ZENECA LIMITED (GB) 1990-11-07 EP disclosed