SCHEMBL9340328

SCHEMBL9340328

O=c1c(Br)c(C(F)(F)F)ncn1-c1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 4/20 0.42
CYP3A4 P08684 4/20 0.42
TSHR P16473 2/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
HIF1A Q16665 1/20 0.42
TXNRD1 Q16881 1/20 0.42
TXNRD3 Q86VQ6 1/20 0.42
TXNRD2 Q9NNW7 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PLK1 P53350 1/20 0.38
PTPN5 P54829 1/20 0.37
MAPT P10636 5/20 0.37
MAPK1 P28482 4/20 0.37
LMNA P02545 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9723134 0.93 POLB (0.40) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9340200 0.92 TDP1 (0.44) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9340421 0.85 CYP3A4 (0.52) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9339513 0.82 ALDH1A1 (0.47) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9340204 0.80 HCAR1 (0.30)
SCHEMBL9339495 0.79 GABRA2 (0.40)
SCHEMBL9723076 0.79 TDP1 (0.45) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9723126 0.78 TDP1 (0.44) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9339503 0.78 TDP1 (0.44) ALDH1A1TDP1CYP3A4TSHRHPGD
SCHEMBL9723045 0.77 HCAR1 (0.36) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0338686-B1 Pyrimidinone derivatives ZENECA LTD (GB) 1994-06-22 EP disclosed
US-5149810-A Chemical intermediates for insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-09-22 US disclosed
US-5077297-A Insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-31 US disclosed
EP-0338686-A2 Pyrimidinone derivatives ZENECA LIMITED (GB) 1989-10-25 EP disclosed