SCHEMBL9345949

SCHEMBL9345949

O=C(CCc1ccc(O)c(O)c1)N1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 9/20 0.56
CACNA1B Q00975 9/20 0.56
CACNB1 Q02641 9/20 0.56
CACNA1C Q13936 7/20 0.56
CACNA1H O95180 1/20 0.56
USP2 O75604 1/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPK1 P28482 1/20 0.53
NPC1 O15118 1/20 0.52
CACNA1G O43497 4/20 0.52
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4904835 0.84 NAAA (0.68) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1H
SCHEMBL16598967 0.82 CACNA2D1 (0.59) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1H
SCHEMBL9346942 0.80 MEN1 (0.57) ALDH1A1MAPK1NPC1KMT2A
SCHEMBL9345400 0.79 NPC1 (0.61) ALDH1A1MAPK1NPC1KMT2A
SCHEMBL9346536 0.78 IAPP (0.53) NPC1KMT2A
SCHEMBL2293693 0.78 CACNA1C (0.69) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1H
SCHEMBL9350110 0.77 NPC1 (0.59) ALDH1A1MAPK1NPC1KMT2A
SCHEMBL10483827 0.75 GAA (0.52) NPC1
SCHEMBL9336419 0.75 FKBP1A (0.64) ALDH1A1MAPK1NPC1KMT2A
SCHEMBL6162758 0.74 CACNA1G (0.85) CACNA2D1CACNA1BCACNB1CACNA1CCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0333522-B1 Catechol derivatives and pharmaceutical preparations containing same MITSUI TOATSU CHEMICALS (JP) 1994-08-17 EP disclosed
US-5232923-A Stimulates production of nerve growth factor; administering for treatment of regressive disorders of the central nervous system MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1993-08-03 US disclosed
EP-0333522-A2 Catechol derivatives and pharmaceutical preparations containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1989-09-20 EP disclosed