SCHEMBL934633

SCHEMBL934633

CC(Cc1cccc(O)c1)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 1/20 0.49
ENPP2 Q13822 1/20 0.48
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
PKM P14618 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
MAPK1 P28482 1/20 0.44
HPGDS O60760 2/20 0.44
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
OPRM1 P35372 2/20 0.43
OPRD1 P41143 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658555 0.84 GRIA2 (0.54) GRIA2ENPP2KDM4ELMNAOPRM1
SCHEMBL2498139 0.84 GRIA2 (0.54) GRIA2ENPP2KDM4ELMNAOPRM1
SCHEMBL17211514 0.84 GRIA2 (0.50) GRIA2ENPP2DRD2DRD1TAAR1
SCHEMBL3654636 0.84 GRIA2 (0.54) GRIA2ENPP2KDM4ELMNAOPRM1
SCHEMBL24915424 0.83 POLB (0.47) TAAR1KDM4EKMT2AMAPTPARP1
SCHEMBL28662062 0.83 ADRB2 (0.45)
SCHEMBL9989813 0.81 SLC1A1 (0.55) TAAR1ALOX15PARP1
SCHEMBL933328 0.81 CYP1A2 (0.47) CYP1A2LMNAPMP22HIF1A
SCHEMBL31324833 0.81 PNMT (0.64) TAAR1KDM4EPARP1CTBP2
SCHEMBL24709885 0.80 ANPEP (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed