SCHEMBL934635

SCHEMBL934635

NC(=O)CCCc1cccc(O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.59
DRD2 P14416 1/20 0.58
DRD1 P21728 1/20 0.58
TAAR1 Q96RJ0 1/20 0.58
MGLL Q99685 1/20 0.53
ENPP2 Q13822 1/20 0.52
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
CALM1 P0DP23 1/20 0.47
IDO1 P14902 1/20 0.47
OPRK1 P41145 1/20 0.47
MAPK1 P28482 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
PKM P14618 1/20 0.47
ALOX15 P16050 1/20 0.47
NFKB1 P19838 1/20 0.47
KMT2A Q03164 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1617652 0.91 DRD2 (0.60) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL3717612 0.85 HDAC6 (0.66) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL31170733 0.85 HDAC6 (0.52) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL19932503 0.84 HDAC6 (0.58) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL11232474 0.82 DRD2 (0.68) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL31674607 0.82 DRD2 (0.68) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL28368586 0.82 DRD2 (0.68) HDAC6DRD2DRD1TAAR1MGLL
SCHEMBL15272646 0.81 MAOA (0.55) HDAC6MAPK1CYP1A2HDAC3ADRA1A
SCHEMBL2762061 0.81 MAPT (0.55) HDAC6MAPTHDAC1HDAC2
SCHEMBL2761735 0.81 MAPT (0.55) HDAC6MAPTHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed
EP-1633715-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS Pfizer Limited (GB) 2006-03-15 EP disclosed
WO-2004108676-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS PFIZER LIMITED (GB) 2004-12-16 WO disclosed