Indoximod

Indoximod

SCHEMBL934800

Cn1cc(C[C@@H](N)C(=O)O)c2ccccc21

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

MLST8MTORRPTOR

The experimentally established mechanism targets of Indoximod. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.71
ALDH1A1 P00352 1/20 0.71
RECQL P46063 1/20 0.71
GPR84 Q9NQS5 1/20 0.54
HTR2A P28223 1/20 0.53
KDM4E B2RXH2 4/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 1/20 0.50
MPO P05164 1/20 0.50
TSHR P16473 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
ARG1 P05089 1/20 0.49
CMA1 P23946 2/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CA2 P00918 1/20 0.49
SCN9A Q15858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(L)-1-Methyltryptophan SCHEMBL19993 1.00 MAPT (0.71) MAPTALDH1A1RECQLGPR84HTR2A
1-Methyltryptophan SCHEMBL14202956 1.00 MAPT (0.71) MAPTALDH1A1RECQLGPR84HTR2A
Indoximod SCHEMBL29349777 1.00 MAPT (0.71) MAPTALDH1A1RECQLGPR84HTR2A
1-Methyltryptophan SCHEMBL19992 1.00 MAPT (0.71) MAPTALDH1A1RECQLGPR84HTR2A
Indoximod SCHEMBL23668055 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A
Indoximod SCHEMBL18395435 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A
Indoximod SCHEMBL30025427 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A
1-Methyltryptophan SCHEMBL23668056 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A
1-Methyltryptophan SCHEMBL20137858 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A
(L)-1-Methyltryptophan SCHEMBL31387967 0.99 MAPT (0.69) MAPTALDH1A1RECQLGPR84HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1893 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122057015-A Cell therapeutic preparation based on tumor specific antigen and application of cell therapeutic preparation in solid tumor 臻辉生物技术(河南)有限公司 2026-05-19 CN claimed
WO-2026090266-A2 IONIZABLE LIPID PRODRUG COMPOUNDS AND LIPID NANOPARTICLES (LNPS) COMPRISING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2026-04-30 WO claimed
US-20260069538-A1 CXCR4 ANTAGONIST LOADED LIPOSOMES AND SILICASOMES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-03-12 US claimed
US-20260049115-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER WITH ECM-AFFINITY PEPTIDES LINKED TO CYTOKINES THE UNIVERSITY OF CHICAGO (US) 2026-02-19 US claimed
US-12539338-B2 Nano-enabled immunotherapy in cancer THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-02-03 US claimed
US-12527872-B2 PEGylated ICD inducer-IDO inhibitor nanoconjugate, and preparation method and use thereof SHANDONG UNIVERSITY (CN) 2026-01-20 US claimed
CN-120154735-A Polyamino acid composite material, preparation method thereof and anti-tumor drug 中国科学院长春应用化学研究所 2025-06-17 CN claimed
US-12280047-B2 Treatment of aneurysms GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2025-04-22 US claimed
CN-119591587-A EGFR dependent small molecule conjugate-1, 3, 4, preparation method and application thereof 江苏省中国科学院植物研究所 2025-03-11 CN claimed
CN-116251062-B Preparation method and application of bacterial membrane-liposome drug-loading system 南通大学 2024-12-17 CN claimed
WO-2011007135-A1 USE OF PRO-INFLAMMATORY COMPOUNDS FOR PROMOTING BONE FORMATION IMPERIAL INNOVATIONS LIMITED (GB) 2011-01-20 WO claimed
EP-2177601-A1 Antigen-presenting cell populations and their use as reagents for enhancing or reducing immune tolerance Medical College of Georgia Research Institute, Inc (US) 2010-04-21 EP claimed
US-7598287-B2 Use of inhibitors of indoleamine-2,3-dioxygenase in combination with other therapeutic modalities MEDICAL COLLEGE OF GEORGIA RESEARCH INSTITUTE, INC. (US) 2009-10-06 US claimed
US-20090123420-A1 Regulation of T Cell-Mediated Immunity by D Isomers of Inhibitors of Indoleamine-2,3-Dioxygenase MEDICAL COLLEGE OF GEORGIA RESEARCH INSTITUTE, INC (US) 2009-05-14 US claimed
US-20090081155-A1 Use of Inhibitors of Indoleamine-2,3-Dioxygenase in Combination with Other Therapeutic Modalities MEDICAL COLLEGE OF GEORGIA RESEARCH INSTITUTE, INC (US) 2009-03-26 US claimed
EP-1501918-A4 ANTIGEN-PRESENTING CELL POPULATIONS AND THEIR USE AS REAGENTS FOR ENHANCING OR REDUCING IMMUNE TOLERANCE MED COLLEGE GEORGIA RES INST (US) 2006-03-29 EP claimed
US-20050186289-A1 Regulation of T cell-mediated immunity by D isomers of inhibitors of indoleamine-2,3-dioxygenase MEDICAL COLLEGE OF GEORGIA RESEARCH INSTITUTE, INC. (US) 2005-08-25 US claimed
EP-1501918-A1 ANTIGEN-PRESENTING CELL POPULATIONS AND THEIR USE AS REAGENTS FOR ENHANCING OR REDUCING IMMUNE TOLERANCE Medical College Of Georgia Research Institute, Inc. (US) 2005-02-02 EP claimed
WO-2003087347-A1 ANTIGEN-PRESENTING CELL POPULATIONS AND THEIR USE AS REAGENTS FOR ENHANCING OR REDUCING IMMUNE TOLERANCE MEDICAL COLLEGE OF GEORGIA RESEARCH INSTITUTE, INC. (US) 2003-10-23 WO claimed
US-20030194803-A1 Antigen-presenting cell populations and their use as reagents for enhancing or reducing immune tolerance NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-10-16 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12539338-B2 Nano-enabled immunotherapy in cancer IDO1, IDO2, BID MAPT 2693/4885ALDH1A1 1966/4885RECQL 1045/4885
US-12280047-B2 Treatment of aneurysms KYNU, HAAO, HCAR2 MAPT 3308/4885ALDH1A1 553/4885RECQL 1635/4885
US-20260049115-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER WITH ECM-AFFINITY PEPTIDES LINKED TO CYTOKINES FN1, MATR3, COL14A1 MAPT 2107/4885ALDH1A1 3744/4885RECQL 4001/4885
US-12527872-B2 PEGylated ICD inducer-IDO inhibitor nanoconjugate, and preparation method and use thereof IDO1, IDO2, TDO2 MAPT 1624/4885ALDH1A1 389/4885RECQL 4476/4885
US-20260069538-A1 CXCR4 ANTAGONIST LOADED LIPOSOMES AND SILICASOMES CXCL12, CXCR4, CXCR5 MAPT 3565/4885ALDH1A1 3405/4885RECQL 2857/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.