SCHEMBL9348598

SCHEMBL9348598

COc1cc(N)c(COCc2ccccc2)c(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
ALOX5 P09917 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP19A1 P11511 1/20 0.39
G6PD P11413 1/20 0.38
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9352506 0.82 TSHR (0.44) TSHRALOX5NPC1RAB9AG6PD
SCHEMBL9352494 0.82 TSHR (0.44) TSHRALOX5G6PDMGAMGAA
SCHEMBL9348656 0.82 TSHR (0.44) TSHRALOX5G6PDMGAMGAA
SCHEMBL9348570 0.78 CYP3A4 (0.37) NPC1CYP19A1POLBTUBB4ATUBB
SCHEMBL9349810 0.77 TSHR (0.48) TSHRALOX5CYP19A1
SCHEMBL9352610 0.77 CTSV (0.48) NPC1RAB9AGAASMN1; SMN2TUBB4A
SCHEMBL30963209 0.75 ALDH1A1 (0.61) TSHRALOX5GAA
SCHEMBL2032107 0.75 ALDH1A1 (0.61) TSHRALOX5GAA
SCHEMBL8864476 0.72 PTGS2 (0.50) NPC1CYP19A1POLBTUBB4ATUBB
SCHEMBL9348434 0.72 CYP19A1 (0.42) TSHRALOX5CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed