SCHEMBL9348570

SCHEMBL9348570

COCOCc1c(N)cc(OC)c(OC)c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
PDE1A P54750 1/20 0.37
PDE1B Q01064 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE1C Q14123 1/20 0.37
PDE3A Q14432 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
CYP19A1 P11511 1/20 0.36
PTGS2 P35354 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
ACHE P22303 1/20 0.34
NPC1 O15118 1/20 0.34
TUBB4A P04350 4/20 0.34
TUBB P07437 4/20 0.34
TUBA3C P0DPH7 4/20 0.34
TUBA1B P68363 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9348493 0.80 CA1 (0.38) CYP3A4MAPTHTR2APTGS2POLB
SCHEMBL9348405 0.80 CYP3A4 (0.37) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL9349736 0.80 CYP3A4 (0.37) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL9348598 0.78 TSHR (0.44) CYP19A1POLBNPC1TUBB4ATUBB
SCHEMBL8864476 0.77 PTGS2 (0.50) CYP3A4MAPTPDE1APDE1BPDE3B
SCHEMBL9348359 0.77 ALDH1A1 (0.41) CYP3A4MAPTTUBB4ATUBBTUBA3C
SCHEMBL9348386 0.74 ALDH1A1 (0.41) CYP3A4MAPTPTGS2KDM4ETUBB4A
SCHEMBL8707967 0.74 FYN (0.42) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL9348470 0.69 ACHE (0.48) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL5838937 0.69 ACHE (0.47) MAPTPDE3AACHETUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed