SCHEMBL9366994

SCHEMBL9366994

O=C(O)NC(CN1CNc2ccccc21)c1nnn[nH]1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
EPHX2 P34913 1/20 0.31
HSD17B3 P37058 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9366970 1.00 ATM (0.32) ATMMEN1KMT2AHDAC2HDAC8
SCHEMBL6693798 0.72 EPHX2 (0.38) ATMMEN1KMT2AHDAC2HDAC8
SCHEMBL5908164 0.72 CYP1A2 (0.45) ALDH1A1
SCHEMBL7650386 0.70 CNR2 (0.42) MEN1KMT2AALDH1A1TSHR
SCHEMBL31285850 0.68 KMT2A (0.42) MEN1KMT2AEPHX2HSD17B3ALDH1A1
SCHEMBL8793695 0.68 KMT2A (0.42) MEN1KMT2AEPHX2HSD17B3ALDH1A1
SCHEMBL6690571 0.68 BRPF1 (0.35) MEN1KMT2AHDAC2HDAC8HDAC6
SCHEMBL6175819 0.65 PTGS1 (0.42) HDAC2HDAC8HDAC6EPHX2HSD17B3
SCHEMBL7413032 0.64 MMP1 (0.36) MEN1KMT2AALDH1A1TSHR
SCHEMBL7417802 0.64 SMN1; SMN2 (0.51) MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449523-B1 Mercapto- or acylthio-trifluoromethyl amide derivatives and their use SQUIBB & SONS INC (US) 1994-08-17 EP disclosed