SCHEMBL9367665

SCHEMBL9367665

C1=C(c2nccs2)CCC(CCN2CCN(c3ccccn3)CC2)C1

nearest known ligand 0.75

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.53
DRD2 P14416 5/20 0.51
DRD3 P35462 4/20 0.51
HTR1A P08908 2/20 0.48
DRD4 P21917 2/20 0.47
HTR2A P28223 1/20 0.47
HTR7 P34969 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9368439 0.86 DRD2 (0.54) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9371451 0.85 DRD2 (0.56) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9367275 0.84 DRD2 (0.55) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9367644 0.82 DRD3 (0.55) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9367241 0.76 DRD2 (0.45) HTR2CDRD2DRD3DRD4HTR2A
SCHEMBL8470779 0.75 DRD2 (0.65) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9367707 0.74 DRD2 (0.51) HTR2CDRD2DRD3DRD4HTR2A
SCHEMBL9370055 0.73 DRD2 (0.49) HTR2CDRD2DRD4HTR2A
SCHEMBL9202816 0.73 DRD2 (0.55) HTR2CDRD2DRD3HTR1ADRD4
SCHEMBL9195812 0.72 DRD2 (0.61) HTR2CDRD2DRD3HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP claimed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431579-B1 Substituted cyclohexenes as central nervous system agents WARNER LAMBERT CO (US) 1994-07-27 EP disclosed
EP-0431579-A2 Substituted cyclohexenes as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4975445-A Antidepressants WARNER-LAMBERT COMPANY (US) 1990-12-04 US disclosed