SCHEMBL9375898

SCHEMBL9375898

CC(=O)Nc1cc(Cl)cn(C2=NC(C)(C)Oc3ccc(C#N)cc32)c1=O

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 11/20 0.37
DRD2 P14416 3/20 0.34
DRD3 P35462 3/20 0.34
EGLN2 Q96KS0 1/20 0.34
BACE1 P56817 1/20 0.32
DYRK1A Q13627 1/20 0.32
KDM4E B2RXH2 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378613 0.89 ABCC9 (0.33) ABCC9DRD2DRD3EGLN2BACE1
SCHEMBL9372276 0.86 ABCC9 (0.34) ABCC9DRD2DRD3EGLN2DYRK1A
SCHEMBL9371959 0.85 EGLN2 (0.39) ABCC9DRD2DRD3EGLN2AR
SCHEMBL9372600 0.85 ABCC9 (0.39) ABCC9
SCHEMBL9377305 0.83 ABCC9 (0.38) ABCC9BACE1
SCHEMBL8088696 0.83 PDE4A (0.37) ABCC9DRD2DRD3EGLN2KDM4E
SCHEMBL9376786 0.82 DRD2 (0.37) ABCC9DRD2DRD3EGLN2DYRK1A
SCHEMBL8084526 0.82 ABCC9 (0.36) ABCC9DRD2DRD3EGLN2KDM4E
SCHEMBL9372773 0.81 DRD2 (0.41) ABCC9DRD2DRD3EGLN2BACE1
SCHEMBL9372978 0.80 VCAM1 (0.38) ABCC9AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371312-B1 Benzoxazine derivatives MERCK PATENT GMBH (DE) 1994-07-20 EP disclosed
US-5036068-A Cardiovascular disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-07-30 US disclosed
EP-0371312-A1 Benzoxazine derivatives MERCK PATENT GmbH (DE) 1990-06-06 EP disclosed