SCHEMBL9378249

SCHEMBL9378249

CCCCCCCCCCCCn1ccnc1C(CCCC)(OCCN(C)C)c1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.37
THRA P10827 2/20 0.32
THRB P10828 2/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 3/20 0.32
HTR1A P08908 2/20 0.32
HTR7 P34969 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
PKM P14618 1/20 0.30
CYP2C19 P33261 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4911325 0.96 TLR8 (0.37) TLR8THRATHRBHTR2AHTR2C
SCHEMBL4902316 0.92 TLR8 (0.33) TLR8CYP1A2CYP3A4CYP2C9PKM
SCHEMBL4910196 0.78 TLR8 (0.42) TLR8HTR2AHTR2CHTR2BHTR1A
SCHEMBL4900357 0.74 ALDH1A1 (0.39) TLR8HTR2AHTR2CHTR1AHTR7
SCHEMBL5616111 0.71 TLR8 (0.37) TLR8THRATHRBHTR2AHTR2C
SCHEMBL9373850 0.69 SIGMAR1 (0.31) THRATHRBHTR2AHTR2CALDH1A1
SCHEMBL9374550 0.69 KDM4E (0.35) HTR2AHTR2CHTR7CYP2C19KMT2A
SCHEMBL4902326 0.69 KMT2A (0.32) CYP1A2CYP3A4CYP2C19ALDH1A1POLB
SCHEMBL4905621 0.68 FYN (0.37) SMN1; SMN2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4904538 0.68 PRKCG (0.34) TLR8THRBHTR2AHTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289380-B1 Aryl-heteroaryl-carbinol derivatives having an analgesic activity ESTEVE LABOR DR (ES) 1994-12-28 EP claimed