SCHEMBL9378692

SCHEMBL9378692

COc1cccc2c1O[C]C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
PTGS2 P35354 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
KDM4E B2RXH2 2/20 0.36
HTR2A P28223 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR7 P34969 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4648888 0.82 MAOB (0.38) PTGS2ALDH1A1MAPTHPGDKDM4E
SCHEMBL2378171 0.69 LMNA (0.60) ALDH1A1MAPTKDM4ELMNA
SCHEMBL5785526 0.68 PARP1 (0.47) CA12CA1CA2CA4CA7
SCHEMBL7516624 0.66 ACHE (0.43) ALDH1A1MAPTHPGDDRD2DRD3
SCHEMBL11106287 0.66 TERT (0.38) CA12CA1CA2CA4CA7
SCHEMBL30465990 0.66 ACHE (0.43) ALDH1A1MAPTHPGDDRD2DRD3
SCHEMBL4140771 0.66 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL13799415 0.66 PARP1 (0.51) ALDH1A1HPGDDRD2DRD3KDM4E
SCHEMBL10800882 0.64 KMT2A (0.40) ALDH1A1DRD2DRD3LMNAHTR5A
SCHEMBL4224918 0.64 HTR7 (0.43) CA12CA1CA2CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0428437-B1 1,2-Benzisoxazole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1994-08-17 EP disclosed
EP-0428437-A1 1,2-Benzisoxazole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-05-22 EP disclosed