SCHEMBL9380385

SCHEMBL9380385

COc1cccc([C@H]2O[C@@H]2/C=C/C=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 3/20 0.41
NPC1 O15118 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HIF1A Q16665 2/20 0.41
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
NFKB1 P19838 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9380409 0.80 MEN1 (0.37) MEN1KMT2ANPC1HTR2CCYP19A1
SCHEMBL9378128 0.80 MEN1 (0.37) MEN1KMT2ANPC1HTR2CCYP19A1
SCHEMBL10372159 0.76 LMNA (0.39) MEN1KMT2ACYP2C19ALDH1A1NFKB1
SCHEMBL9377930 0.76 LMNA (0.39) MEN1KMT2ACYP2C19ALDH1A1NFKB1
SCHEMBL9382305 0.73 HTR2C (0.40) CYP2C19CHRM2HTR2CLMNAHTR2A
SCHEMBL11162641 0.72 HTR2C (0.50) MEN1KMT2AKDM4ENPC1CYP3A4
SCHEMBL3762403 0.68 HTR2C (0.46) MEN1KMT2AKDM4ENPC1CYP3A4
SCHEMBL23676966 0.67 HTR2C (0.61) MEN1KMT2AKDM4ENPC1CYP3A4
SCHEMBL9692360 0.67 TSHR (0.51) MEN1KMT2AKDM4ENPC1CYP3A4
SCHEMBL25259513 0.66 RELA (0.62) RELACHRM2CHRM1CHRM3CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335315-B1 New alkanephenones CIBA GEIGY AG (CH) 1994-06-22 EP disclosed
US-5149717-A Alkanophenones useful for treating allergies CIBA-GEIGY CORPORATION (US) 1992-09-22 US disclosed
EP-0335315-A1 New alkanephenones CIBA-GEIGY AG (CH) 1989-10-04 EP disclosed