SCHEMBL9384334

SCHEMBL9384334

O=C(Cc1ccccc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.68
CES2 O00748 2/20 0.68
FNTA P49354 1/20 0.52
FNTB P49356 1/20 0.52
AKR1B1 P15121 1/20 0.50
CNR2 P34972 1/20 0.50
F2 P00734 1/20 0.47
CNR1 P21554 2/20 0.46
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28577864 0.79 CES1 (0.54) CES1CES2FNTAFNTBAKR1B1
SCHEMBL4642302 0.79 POLB (0.48) CES1CES2CNR2CNR1TDP1
Phenylpyruvate SCHEMBL27787637 0.79 CES1 (0.73) CES1CES2FNTAFNTBAKR1B1
Phenylpyruvate SCHEMBL43235 0.78 CES1 (0.80) CES1CES2FNTAFNTBAKR1B1
Phenylpyruvate SCHEMBL28203540 0.78 CES1 (0.80) CES1CES2FNTAFNTBAKR1B1
SCHEMBL574185 0.78 CES1 (1.00) CES1CES2FNTAFNTBAKR1B1
SCHEMBL451546 0.78 CES1 (0.64) CES1CES2FNTAFNTBAKR1B1
SCHEMBL4641484 0.78 TDP1 (0.47) CES1CES2CNR2CNR1TDP1
Phenylpyruvate SCHEMBL11193388 0.76 CES1 (0.76) CES1CES2FNTAFNTBAKR1B1
Phenylpyruvate SCHEMBL468389 0.76 CES1 (0.76) CES1CES2FNTAFNTBAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0376197-B1 Sulfur-containing heterocyclic compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-10-12 EP disclosed
US-5071841-A For prevention of bone reabsorption TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-12-10 US disclosed
EP-0376197-A1 Sulfur-containing heterocyclic compounds Takeda Chemical Industries, Ltd. (JP) 1990-07-04 EP disclosed