SCHEMBL9389023

SCHEMBL9389023

CC(C)c1cccc2c(=O)cc(O)c(=O)[nH]c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 9/20 0.45
DDO Q99489 5/20 0.45
KDM4E B2RXH2 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
PLA2G7 Q13093 3/20 0.42
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CYP3A4 P08684 2/20 0.39
HPGD P15428 2/20 0.39
MDM4 O15151 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
TYR P14679 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
CA5A P35218 1/20 0.39
HTT P42858 1/20 0.39
HDAC4 P56524 1/20 0.39
MDM2 Q00987 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583717 0.80 DAO (0.66) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9390027 0.77 DAO (0.68) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9389395 0.76 KDM4E (0.46) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9389416 0.76 DAO (0.66) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9388997 0.76 DAO (0.66) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9393346 0.76 DAO (0.49) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9389819 0.76 KIF11 (0.47) DAODDOKDM4ETDP1PLA2G7
SCHEMBL9389042 0.76 DAO (0.36) DAODDOTRPV1
SCHEMBL9392651 0.76 DAO (0.49) DAODDOKDM4ETDP1CA1
SCHEMBL9387636 0.74 DAO (0.55) DAODDOKDM4ETDP1PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed