SCHEMBL9389819

SCHEMBL9389819

CC(C)(C)c1cccc2c(=O)cc(O)c(=O)[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
DAO P14920 8/20 0.45
DDO Q99489 5/20 0.45
TDP1 Q9NUW8 2/20 0.43
PLA2G7 Q13093 4/20 0.43
HDAC4 P56524 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
CA2 P00918 1/20 0.39
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583717 0.80 DAO (0.66) KDM4EALDH1A1LMNAPOLBHPGD
SCHEMBL9390027 0.77 DAO (0.68) KDM4EALDH1A1LMNADAODDO
SCHEMBL9389416 0.76 DAO (0.66) KDM4EDAODDOTDP1PLA2G7
SCHEMBL9389395 0.76 KDM4E (0.46) KDM4EDAODDOTDP1PLA2G7
SCHEMBL9393346 0.76 DAO (0.49) KDM4EALDH1A1LMNAHPGDDAO
SCHEMBL9388997 0.76 DAO (0.66) KDM4ELMNADAODDOTDP1
SCHEMBL9389023 0.76 DAO (0.45) KDM4EALDH1A1LMNAHPGDHTT
SCHEMBL9387636 0.74 DAO (0.55) KDM4EALDH1A1LMNAHPGDDAO
SCHEMBL9389330 0.73 KDM4E (0.43) KDM4EDAODDOTDP1PLA2G7
SCHEMBL16154714 0.72 KIF11 (0.54) KIF11KDM4EALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed