SCHEMBL9395751

SCHEMBL9395751

COc1c([N+](=O)[O-])cc(C#N)c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.44
IMPDH1 P20839 1/20 0.44
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 1/20 0.42
VCAM1 P19320 1/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RECQL P46063 1/20 0.41
GRM6 O15303 1/20 0.40
GRIA1 P42261 1/20 0.40
GRIA2 P42262 1/20 0.40
GRIA3 P42263 1/20 0.40
GRIA4 P48058 1/20 0.40
LMNA P02545 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GPR35 Q9HC97 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11720706 0.77 CTSB (0.55) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL9081258 0.77 CTSB (0.51) ALDH1A1TDP1HTTMAPTKDM4E
SCHEMBL6742801 0.75 TDP1 (0.47) ALDH1A1TDP1VCAM1MAPTMEN1
SCHEMBL11948737 0.74 HTT (0.45) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL9736340 0.74 VCAM1 (0.49) ALDH1A1TDP1VCAM1MAPTKDM4E
SCHEMBL16901738 0.74 GPR35 (0.44) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL7373383 0.73 TPMT (0.44) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL30673260 0.73 GPR35 (0.48) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL26927308 0.73 GPR35 (0.48) ALDH1A1TDP1HTTVCAM1MAPT
SCHEMBL1341782 0.73 TDP1 (0.55) IMPDH2IMPDH1ALDH1A1TDP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315959-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-03-02 EP disclosed
US-5026704-A Neuroleptic agent, quisqualate-antagonist NOVO NORDISK A/S (DK) 1991-06-25 US disclosed
US-4948794-A NEUROLEPTIC AGENTS A/S FERROSAN (DK) 1990-08-14 US disclosed
EP-0315959-A2 Quinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1989-05-17 EP disclosed