SCHEMBL9397242

SCHEMBL9397242

NC1(C(=O)O)CCc2c(cccc2N(CCCl)CCCl)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.43
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
CXCR5 P32302 1/20 0.32
PTGER1 P34995 1/20 0.31
PTGER3 P43115 1/20 0.31
PTGIR P43119 1/20 0.31
PTGDR Q13258 1/20 0.31
CYP3A4 P08684 3/20 0.30
ALDH1A1 P00352 2/20 0.30
ALOX15 P16050 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
HIF1A Q16665 2/20 0.30
ABCB11 O95342 1/20 0.30
CHRM2 P08172 1/20 0.30
ADRA2A P08913 1/20 0.30
CHRM1 P11229 1/20 0.30
ACHE P22303 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4600871 0.81 RXRA (0.36) RXRARXRBRXRGCXCR5PTGER1
SCHEMBL4599994 0.76 GRM2 (0.39) ADRA2A
SCHEMBL22852446 0.76 RAD52 (0.31) RAD52PTGER1PTGER3PTGIRPTGDR
SCHEMBL9397128 0.74 RAD52 (0.61) RAD52RXRARXRBRXRGCYP3A4
SCHEMBL4600677 0.74 GABRA1 (0.37) CYP3A4ALDH1A1ALOX15PTGS1TDP1
SCHEMBL4601314 0.73 AKR1C3 (0.36) MEN1KMT2A
SCHEMBL4599719 0.73 CXCR5 (0.36) RXRACXCR5ALDH1A1KDM4ELMNA
SCHEMBL4599810 0.71 ADRA2A (0.47) CHRM2ADRA2ACHRM1ACHEDRD3
SCHEMBL4600670 0.71 RXRA (0.41) RXRARXRBRXRGCXCR5PTGER1
SCHEMBL4599658 0.70 CYP3A4 (0.36) CYP3A4ALDH1A1HIF1APTGS1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5284774-A Antineoplastic, system-L specific amino acid nitrogen mustards THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECY. OF THE DEPT. OF HEALTH & HUMAN RESOURCES (US) 1994-02-08 US disclosed
US-4772632-A REDUCED MYELOSUPPRESSION THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1988-09-20 US disclosed