SCHEMBL9399167

SCHEMBL9399167

CNC(=S)[C@]1(c2ccncc2)CCCC[C@H]1OC(=O)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
BCHE P06276 1/20 0.35
SLC6A3 Q01959 1/20 0.35
LMNA P02545 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.35
CHRNA7 P36544 2/20 0.34
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
HTR3E A5X5Y0 2/20 0.33
HTR3B O95264 2/20 0.33
HTR3A P46098 2/20 0.33
HTR3D Q70Z44 2/20 0.33
HTR3C Q8WXA8 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9399179 1.00 ITGA4 (0.36) ITGA4ITGB7BCHESLC6A3LMNA
SCHEMBL9491327 0.89 CNR2 (0.41) ITGA4ITGB7LMNACYP2D6
SCHEMBL9490368 0.89 CNR2 (0.41) ITGA4ITGB7LMNACYP2D6
SCHEMBL9490471 0.89 CNR2 (0.41) ITGA4ITGB7LMNACYP2D6
SCHEMBL9520161 0.89 CNR2 (0.41) ITGA4ITGB7LMNACYP2D6
SCHEMBL9490420 0.87 CYP2D6 (0.36) ITGA4ITGB7LMNAMAPTCYP2D6
SCHEMBL9521837 0.87 CYP2D6 (0.36) ITGA4ITGB7LMNAMAPTCYP2D6
SCHEMBL9521077 0.84 ALDH1A1 (0.41) ITGA4ITGB7LMNANPSR1MAPT
SCHEMBL9490387 0.84 ALDH1A1 (0.41) ITGA4ITGB7LMNANPSR1MAPT
SCHEMBL9491487 0.82 ITGA4 (0.41) ITGA4ITGB7BCHESLC6A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5342848-A Relaxation of vascular smooth muscle RHONE-POULENC RORER LIMITED (GB) 1994-08-30 US claimed
WO-1991012242-A1 THIOFORMAMIDE DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1991-08-22 WO claimed
US-5342848-A Relaxation of vascular smooth muscle RHONE-POULENC RORER LIMITED (GB) 1994-08-30 US disclosed
EP-0514419-A1 THIOFORMAMIDE DERIVATIVES Aventis Pharma S.A. (FR) 1992-11-25 EP disclosed
WO-1991012242-A1 THIOFORMAMIDE DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1991-08-22 WO disclosed