SCHEMBL9400876

SCHEMBL9400876

O=C1c2cc(F)ccc2S(=O)(=O)N1CCCBr

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
CA9 Q16790 8/20 0.47
CA12 O43570 7/20 0.47
RAB9A P51151 2/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
CA2 P00918 2/20 0.45
CA1 P00915 2/20 0.45
NPC1 O15118 1/20 0.41
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
HTR7 P34969 1/20 0.40
HTR6 P50406 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8667503 0.96 ADRA1D (0.51) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8667501 0.81 ADRA1D (0.39) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8973563 0.79 CA9 (0.72) CA9CA12HPGDCA2HTR1A
SCHEMBL7815416 0.79 ADRA1D (0.51) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8667643 0.79 CA9 (0.51) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8670252 0.76 ADRA1D (0.53) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8047945 0.76 CA9 (0.42) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8671286 0.75 HDAC1 (0.55) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL6324557 0.75 CA9 (0.73) ADRA1DADRA1AADRA1BCA9CA12
SCHEMBL8047906 0.74 CA9 (0.49) ADRA1DADRA1AADRA1BCA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314884-A Antidepressants, anxiolytic agents TROPONWERKE GMBH & CO. (DE) 1994-05-24 US disclosed
US-5187276-A Anxiolytics, neuroleptics, antidepressants, and nootropic agents TROPONWERKE GMBH & CO. KG. (DE) 1993-02-16 US disclosed
US-4988809-A CENTRAL NERVOUS SYSTEM TROPONWERKE GMBH & CO., KG (DE) 1991-01-29 US disclosed
US-4937343-A NEUROLEPTICS OR ANTIDEPRESSANTS TROPONWERKE GMBH & CO. KG (DE) 1990-06-26 US disclosed