SCHEMBL9401128

SCHEMBL9401128

CCC(=O)NCCc1c(Cc2ccc(OC)cc2)[nH]c2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.64
MTNR1B P49286 6/20 0.64
CYP2C19 P33261 3/20 0.64
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
HPGD P15428 2/20 0.64
TSHR P16473 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
ALDH1A1 P00352 1/20 0.64
CYP2D6 P10635 1/20 0.64
MAPT P10636 1/20 0.64
ALOX15 P16050 1/20 0.64
MEN1 O00255 2/20 0.62
CYP2C9 P11712 2/20 0.62
KMT2A Q03164 2/20 0.62
KDM4E B2RXH2 1/20 0.52
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9751553 0.89 MTNR1A (0.79) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL9401112 0.89 MTNR1A (0.79) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL29138489 0.85 MTNR1A (0.60) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL7692306 0.81 KDM4E (0.56) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL30669507 0.80 KDM4E (0.48) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL29138480 0.80 ALB (0.51) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL29138474 0.80 ALB (0.51) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL9401123 0.79 KDM4E (0.44) MTNR1AMTNR1BCYP2C19ALDH1A1MEN1
SCHEMBL29138500 0.78 MTNR1A (0.88) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4
SCHEMBL30669508 0.78 MTNR1A (0.88) MTNR1AMTNR1BCYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314908-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1994-05-24 US disclosed
EP-0549916-A2 Compounds useful as antiproliferative agents WHITBY RESEARCH, Inc. (US) 1993-07-07 EP disclosed
US-5206377-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1993-04-27 US disclosed