SCHEMBL9401112

SCHEMBL9401112

CCC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.79
MTNR1B P49286 5/20 0.79
TDP1 Q9NUW8 3/20 0.79
CYP1A2 P05177 2/20 0.79
CYP3A4 P08684 2/20 0.79
HPGD P15428 2/20 0.79
TSHR P16473 2/20 0.79
CYP2C19 P33261 2/20 0.79
MAPT P10636 2/20 0.79
ALOX15 P16050 2/20 0.79
ALDH1A1 P00352 1/20 0.79
CYP2D6 P10635 1/20 0.79
MEN1 O00255 1/20 0.78
CYP2C9 P11712 1/20 0.78
KMT2A Q03164 1/20 0.78
CHRNB2 P17787 1/20 0.52
CHRNA7 P36544 1/20 0.52
CHRNA4 P43681 1/20 0.52
EGFR P00533 1/20 0.52
SRC P12931 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401128 0.89 MTNR1A (0.64) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL1626901 0.89 MTNR1A (1.00) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
Luzindole SCHEMBL4869000 0.88 MTNR1A (1.00) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL9401161 0.80 MTNR1A (0.84) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL28134995 0.79 TDP1 (0.52) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
Luzindole SCHEMBL9118261 0.79 MEN1 (0.81) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL2944735 0.78 MTNR1A (0.66) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL2087168 0.77 HPGD (0.61) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL9751553 0.77 MTNR1A (0.79) MTNR1AMTNR1BTDP1CYP1A2CYP3A4
SCHEMBL8001497 0.76 MTNR1A (0.63) MTNR1AMTNR1BTDP1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314908-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1994-05-24 US disclosed
EP-0549916-A2 Compounds useful as antiproliferative agents WHITBY RESEARCH, Inc. (US) 1993-07-07 EP disclosed
US-5206377-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1993-04-27 US disclosed