SCHEMBL9405535

SCHEMBL9405535

O=[N+]([O-])c1ccc(Oc2ccccc2-c2ccc(CCBr)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
HSPB1 P04792 2/20 0.42
PTGS2 P35354 1/20 0.42
CYP19A1 P11511 2/20 0.41
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
FFAR4 Q5NUL3 2/20 0.41
KCNH2 Q12809 4/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
MAPT P10636 3/20 0.40
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
KCNJ1 P48048 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331117 0.90 HSPB1 (0.44) HSPB1PTGS2CYP19A1CYP11B1CYP11B2
SCHEMBL27386744 0.86 MAPT (0.46) HSPB1CYP19A1CYP11B1CYP11B2MAPT
SCHEMBL8444172 0.82 NCOA1 (0.58) HSPB1PTGS2FFAR4NCOA1NCOA3
SCHEMBL8332373 0.80 ACHE (0.51) HSPB1PTGS2FFAR4NCOA1NCOA3
SCHEMBL9812692 0.79 ADRA2A (0.50) HSPB1PTGS2CYP19A1CYP11B1CYP11B2
SCHEMBL9087468 0.79 HSPB1 (0.59) HSPB1MAPTALDH1A1KDM4EMEN1
SCHEMBL27324556 0.79 MEN1 (0.47) HSPB1CYP19A1CYP11B1CYP11B2MAPT
Water SCHEMBL11780560 0.78 ADRA2A (0.49) HSPB1PTGS2CYP19A1CYP11B1CYP11B2
SCHEMBL9405534 0.78 ADRA2A (0.47) HSPB1PTGS2FFAR4NCOA1NCOA3
SCHEMBL8444830 0.77 PTGS2 (0.47) HSPB1PTGS2FFAR4KCNH2NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5310737-A Benzo-fused lactams that promote the release of growth hormone MERCK & CO., INC. (US) 1994-05-10 US disclosed