SCHEMBL9428138

SCHEMBL9428138

Cc1ccc2c(c1)C(=O)N(C)C(c1ccc(C(C)(C)C)cc1)C2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
METAP1 P53582 2/20 0.36
TSHR P16473 1/20 0.35
RIPK1 Q13546 1/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
USP2 O75604 1/20 0.34
CHRNA7 P36544 1/20 0.33
NR1I2 O75469 2/20 0.33
HDAC4 P56524 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
PTAFR P25105 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9407110 0.86 PBRM1 (0.37) RIPK1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8782099 0.83 HTR2A (0.44) ACHEHTR2AHTR2CHTR2BHDAC1
SCHEMBL9427669 0.77 TSHR (0.38) TSHRRIPK1USP2
SCHEMBL28922654 0.72 ACHE (0.50) ACHEHTR2AHTR2CHTR2BMETAP1
SCHEMBL28922605 0.72 ACHE (0.50) ACHEHTR2AHTR2CHTR2BMETAP1
SCHEMBL10085914 0.70 NPC1 (0.56) TSHRHDAC1HDAC4HDAC6PTAFR
SCHEMBL9429146 0.70 HRH3 (0.36) HTR2AHTR2CRIPK1
SCHEMBL8783196 0.66 ESR1 (0.45) ACHEHTR2AHTR2CHTR2BMAPT
SCHEMBL435024 0.65 ACHE (0.45) ACHEHTR2AHTR2CHTR2BMETAP1
SCHEMBL8782370 0.65 DRD2 (0.39) HTR2AHTR2CRIPK1HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5330991-A Tetrahydroisoquinoline compounds and fungicides containing the same TOSOH CORPORATION (JP) 1994-07-19 US disclosed
EP-0528553-A1 Tetrahydroisoquinoline derivatives, processes for producing the same and fungicides containing the same TOSOH CORPORATION (JP) 1993-02-24 EP disclosed