SCHEMBL9409102

SCHEMBL9409102

NC(=O)c1cc(N(F)c2cc(F)c(F)c(F)c2F)c(N(F)c2cc(F)c(F)c(F)c2F)cc1C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.36
CES2 O00748 2/20 0.32
CES1 P23141 2/20 0.32
PRKD3 O94806 1/20 0.30
MAPK9 P45984 1/20 0.30
MAPKAPK2 P49137 1/20 0.30
MAPK10 P53779 1/20 0.30
ROCK1 Q13464 1/20 0.30
ACVR2B Q13705 1/20 0.30
MYLK Q15746 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30
PRKD2 Q9BZL6 1/20 0.30
NLK Q9UBE8 1/20 0.30
PI4KB Q9UBF8 1/20 0.30
ALK Q9UM73 1/20 0.30
MAP2K2 P36507 1/20 0.30
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9409076 0.90 CFTR (0.33) DGAT1
SCHEMBL829400 0.73 DGAT1 (0.45) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL28085635 0.73 DGAT1 (0.45) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL8834688 0.69 GRM5 (0.35) PRKD3
SCHEMBL4345385 0.69
SCHEMBL3026712 0.68 CES2 (0.38) CES2CES1
SCHEMBL12825653 0.68 CES2 (0.31) CES2CES1
SCHEMBL4591061 0.66 DGAT1 (0.42) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL26907499 0.66
SCHEMBL2915007 0.66 CES2 (0.39) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP claimed
EP-0600832-A1 Derivatives of diamino benzoic and diamino phthalic acid und their use as protein linase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP disclosed