SCHEMBL9409485

SCHEMBL9409485

COC(=O)CC[C@H]1CC[C@H](NC(=O)c2ccc(-c3ccncc3)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 12/20 0.51
ROCK1 Q13464 6/20 0.51
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
USP30 Q70CQ3 1/20 0.47
CYP46A1 Q9Y6A2 1/20 0.47
MAPK14 Q16539 2/20 0.47
SMYD3 Q9H7B4 2/20 0.46
HSPB1 P04792 1/20 0.44
CYP2C9 P11712 1/20 0.44
MAPK11 Q15759 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9409446 0.86 MEN1 (0.55) ROCK2ROCK1MEN1NPC1RAB9A
SCHEMBL9233873 0.78 HPGD (0.42) MEN1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL9233868 0.78 HPGD (0.42) MEN1NPC1RAB9AKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL9234972 0.78 ITGB3 (0.46) MEN1KMT2AMAPK14SMYD3CYP2C9
SCHEMBL9409367 0.77 ALDH1A1 (0.46) MAPK14SMYD3CYP2C9
SCHEMBL9415854 0.77 ALDH1A1 (0.46) MAPK14SMYD3CYP2C9
Hydrochloric Acid SCHEMBL9409523 0.76 ALDH1A1 (0.46) MAPK14SMYD3CYP2C9
Hydrochloric Acid SCHEMBL9409352 0.76 ALDH1A1 (0.46) MAPK14SMYD3CYP2C9
Hydrochloric Acid SCHEMBL9409464 0.76 SMYD3 (0.44) MAPK14SMYD3CYP2C9
SCHEMBL9409398 0.76 HTR2A (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604800-A1 4- 4- 4-(carboxyalkyl)-phenyl amino carbonyl -phenyl -piperedines as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-07-06 EP disclosed