SCHEMBL9409997

SCHEMBL9409997

CSc1ncc(CC(=O)O)c(O)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
NTRK1 P04629 1/20 0.38
POLB P06746 3/20 0.36
ALDH1A1 P00352 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AKR1B1 P15121 1/20 0.35
RAB9A P51151 1/20 0.35
ALOX15 P16050 1/20 0.34
RXFP1 Q9HBX9 2/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4276535 0.83 MEN1 (0.53) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL17156365 0.82 MEN1 (0.42) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL9298613 0.80 MEN1 (0.44) MEN1KMT2APOLBALDH1A1TDP1
SCHEMBL31483966 0.77 MEN1 (0.41) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL12639128 0.77 ALDH1A1 (0.43) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL17506379 0.76 NTRK1 (0.39) MEN1KMT2ANTRK1ALDH1A1THRB
SCHEMBL17156348 0.76 DHFR (0.38) MEN1KMT2APOLBALDH1A1TDP1
SCHEMBL2490824 0.75 MEN1 (0.37) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL46639 0.74 MEN1 (0.53) MEN1KMT2ANTRK1POLBALDH1A1
SCHEMBL9785565 0.73 MAPT (0.38) MEN1KMT2APOLBTDP1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed
EP-0612746-A1 Pyrimidines and their pharmaceutical acceptable salts and their use as medicines MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1994-08-31 EP disclosed
US-5264435-A Treatment of neurological diseases MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1993-11-23 US disclosed
US-5147876-A Nervous system disorders MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-09-15 US disclosed
EP-0379806-A2 Pyrimidines and their pharmaceutical acceptable salts, and their use as medicines MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1990-08-01 EP disclosed