SCHEMBL9410787

SCHEMBL9410787

COc1cccc(C(O)C(N)C2Cc3ccc(OCc4ccccc4)c(OCc4ccccc4)c3C2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 13/20 0.44
AGTR1 P30556 2/20 0.44
MAOB P27338 1/20 0.40
ABCB1 P08183 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LRRK2 Q5S007 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540992 0.79 AGTR2 (0.44) AGTR2AGTR1
SCHEMBL8978466 0.78 AGTR2 (0.44) AGTR2AGTR1KMT2ALRRK2
SCHEMBL8549721 0.76 AGTR2 (0.44) AGTR2AGTR1
SCHEMBL8593552 0.74 ADRB3 (0.45) AGTR2
SCHEMBL9410790 0.73 AGTR2 (0.40) AGTR2AGTR1MAOBABCB1HTR1A
SCHEMBL8545450 0.71 AGTR2 (0.40) AGTR2AGTR1DRD2
SCHEMBL8541940 0.68 KDM1A (0.43) AGTR2AGTR1MAOB
SCHEMBL9410814 0.68 MAOB (0.36) AGTR2AGTR1MAOBABCB1HTR1A
SCHEMBL2580244 0.67 MAOB (0.55) MAOBABCB1HTR1ADRD2KMT2A
SCHEMBL30863337 0.66 KMT2A (0.61) MAOBKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608568-A1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID COMPANY (US) 1994-08-03 EP disclosed