SCHEMBL9416807

SCHEMBL9416807

Cc1ccc(-c2c(N)noc2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
PTGS2 P35354 2/20 0.42
PTGS1 P23219 1/20 0.38
HEXA P06865 1/20 0.37
HEXB P07686 1/20 0.37
MAP4K4 O95819 1/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
UBE2N P61088 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
IKBKB O14920 1/20 0.36
MLYCD O95822 2/20 0.36
BRD4 O60885 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416881 0.85 PTGS2 (0.52) ESR1ESR2PTGS2PTGS1KDM4E
SCHEMBL9416820 0.83 PTGS1 (0.43) ESR1ESR2PTGS2PTGS1HEXA
SCHEMBL8765879 0.83 ESR1 (0.56) ESR1ESR2PTGS2PTGS1MAP4K4
SCHEMBL9416851 0.83 MLYCD (0.48) ESR1ESR2PTGS2HEXAHEXB
SCHEMBL10503592 0.73 MLYCD (0.64) MLYCDBRD4ENPP1TDO2
SCHEMBL5324584 0.70 IDO1 (0.37) ALDH1A1BRD4
SCHEMBL8765096 0.70 L3MBTL1 (0.45) ESR1ESR2PTGS2PTGS1MAP4K4
SCHEMBL20837302 0.67 ENPP1 (0.41) HEXAHEXBMEN1KMT2AIKBKB
SCHEMBL19367734 0.66 BRD4 (0.72) HEXAHEXBKDM4EIKBKBMLYCD
SCHEMBL10200524 0.63 MAP4K4 (0.56) PTGS2PTGS1MAP4K4MLYCDBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220947-B1 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO (JP) 1994-06-15 EP claimed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP claimed