SCHEMBL8765879

SCHEMBL8765879

Nc1noc(C(F)(F)F)c1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.56
ESR2 Q92731 1/20 0.56
PTGS1 P23219 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
PTGS2 P35354 3/20 0.50
BRD4 O60885 3/20 0.43
TDO2 P48775 1/20 0.43
POLB P06746 1/20 0.41
GSK3B P49841 1/20 0.41
MLYCD O95822 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 2/20 0.40
AKT2 P31751 1/20 0.40
MAP4K4 O95819 1/20 0.39
NOTUM Q6P988 1/20 0.38
BRD2 P25440 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765096 0.86 L3MBTL1 (0.45) ESR1ESR2PTGS1L3MBTL1PTGS2
SCHEMBL9416881 0.84 PTGS2 (0.52) ESR1ESR2PTGS1L3MBTL1PTGS2
SCHEMBL9416807 0.83 ESR1 (0.43) ESR1ESR2PTGS1L3MBTL1PTGS2
SCHEMBL9416820 0.83 PTGS1 (0.43) ESR1ESR2PTGS1L3MBTL1PTGS2
SCHEMBL11459501 0.73 PTPN1 (0.55) PTGS1L3MBTL1PTGS2BRD4TDO2
SCHEMBL6439781 0.72 ESR1 (1.00) ESR1ESR2PTGS1PTGS2MLYCD
SCHEMBL8784588 0.72 MAP4K4 (0.69) PTGS1PTGS2BRD4TDO2MAPK1
SCHEMBL8764932 0.71 MLYCD (0.63) ESR1ESR2PTGS1L3MBTL1PTGS2
SCHEMBL5698365 0.70 PTGS2 (0.77) ESR1ESR2PTGS1PTGS2
SCHEMBL6248342 0.70 PTGS2 (0.77) ESR1ESR2PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220947-B1 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO (JP) 1994-06-15 EP claimed
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US claimed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP claimed
EP-0375670-B1 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO (JP) 1997-08-06 EP disclosed
EP-0220947-B1 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO (JP) 1994-06-15 EP disclosed
EP-0375670-A2 Process for preparing 3-polyfluoroalkylisoxazolylamines SHIONOGI & CO., LTD. (JP) 1990-06-27 EP disclosed
US-4797492-A INTERMEDIATES FOR BACTERICIDES; HERBICIDES OR FUNGICIDES SHIONOGI & CO., LTD. (JP) 1989-01-10 US disclosed
EP-0220947-A2 Polyfluoroalkylisoxazolylamines, their preparation and use SHIONOGI & CO., LTD. (JP) 1987-05-06 EP disclosed