SCHEMBL9417147

SCHEMBL9417147

Nc1nc(N)c2ncn(OCC(CO)OCP(=O)(O)O)c2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
FGFR1 P11362 3/20 0.41
SLC22A6 Q4U2R8 2/20 0.40
NT5E P21589 1/20 0.39
HPRT1 P00492 7/20 0.38
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
AHCY P23526 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
NFKB1 P19838 1/20 0.34
BLM P54132 1/20 0.34
VCP P55072 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
TYMP P19971 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9417199 0.87 CDK1 (0.39) CYP3A4FGFR1NT5EHPRT1CDK1
SCHEMBL9417190 0.86 CYP3A4 (0.55) CYP3A4FGFR1SLC22A6AHCY
SCHEMBL9555809 0.86 CYP3A4 (0.55) CYP3A4FGFR1SLC22A6AHCY
SCHEMBL9555564 0.86 CYP3A4 (0.55) CYP3A4FGFR1SLC22A6AHCY
SCHEMBL9858340 0.83 HPRT1 (0.43) CYP3A4FGFR1SLC22A6NT5EHPRT1
SCHEMBL29450587 0.82 HPRT1 (0.55) CYP3A4FGFR1SLC22A6HPRT1CDK1
SCHEMBL15516660 0.82 HPRT1 (0.55) CYP3A4FGFR1SLC22A6HPRT1CDK1
SCHEMBL172847 0.82 HPRT1 (0.55) CYP3A4FGFR1SLC22A6HPRT1CDK1
SCHEMBL9555352 0.82 HPRT1 (0.58) CYP3A4HPRT1MEN1ALDH1A1LMNA
SCHEMBL9555507 0.82 HPRT1 (0.58) CYP3A4HPRT1MEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0319228-B1 Novel compounds BEECHAM GROUP PLC (GB) 1994-11-02 EP claimed
US-5247085-A Phosphonate containing purine compounds BEECHAM GROUP P.L.C. (GB) 1993-09-21 US claimed
EP-0319228-B1 Novel compounds BEECHAM GROUP PLC (GB) 1994-11-02 EP disclosed
US-5247085-A Phosphonate containing purine compounds BEECHAM GROUP P.L.C. (GB) 1993-09-21 US disclosed
EP-0319228-A2 Novel compounds BEECHAM GROUP PLC (GB) 1989-06-07 EP disclosed