SCHEMBL9417859

SCHEMBL9417859

C=CCc1cc(C(C)=O)c(OC)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.46
CYP3A4 P08684 5/20 0.46
PTGS1 P23219 2/20 0.46
HTT P42858 1/20 0.42
GABRA1 P14867 3/20 0.42
GABRB2 P47870 3/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
PTPN1 P18031 1/20 0.41
CNR2 P34972 2/20 0.41
TSHR P16473 1/20 0.41
ALOX15 P16050 1/20 0.41
POLB P06746 1/20 0.41
PAX8 Q06710 1/20 0.41
ALDH1A1 P00352 2/20 0.41
AR P10275 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
CA9 Q16790 1/20 0.40
PPARG P37231 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3959266 0.88 HTT (0.60) ALOX5CYP3A4PTGS1HTTGABRA1
SCHEMBL9417934 0.88 PTPN1 (0.52) CYP3A4HTTPTPN1
SCHEMBL9739173 0.86 NR1H4 (0.47) CYP3A4HTTCNR2TSHRALDH1A1
SCHEMBL5339173 0.83 ALOX5 (0.41) ALOX5CYP3A4PTGS1GABRA1GABRB2
SCHEMBL9417761 0.82 NR1H4 (0.42) ALOX5PPARA
SCHEMBL11897974 0.81 CYP3A4 (0.50) CYP3A4HTTTSHRPAX8ALDH1A1
SCHEMBL942820 0.79 ALDH1A1 (0.55) ALOX5CYP3A4PTGS1HTTGABRA1
SCHEMBL29415497 0.79 ALDH1A1 (0.55) ALOX5CYP3A4PTGS1HTTGABRA1
SCHEMBL30880294 0.78 ALOX5 (0.49) ALOX5CYP3A4PTGS1HTTGABRA1
SCHEMBL13596109 0.78 CYP3A4 (0.50) CYP3A4HTTTSHRPAX8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294613-A Benzene derivatives of p-substituted ether and acid or ester ELI LILLY AND COMPANY (US) 1994-03-15 US disclosed
US-5098613-A Aromatic ethers for treatment of mammals ELI LILLY AND COMPANY (US) 1992-03-24 US disclosed
US-4945099-A LEUKOTRIENE ANTAGONIST ELI LILLY AND COMPANY (US) 1990-07-31 US disclosed
EP-0276065-B1 ANTI-INFLAMMATORY AGENTS ELI LILLY AND COMPANY (US) 1990-06-06 EP disclosed
EP-0276065-A1 Anti-inflammatory agents ELI LILLY AND COMPANY (US) 1988-07-27 EP disclosed