SCHEMBL9419052

SCHEMBL9419052

CC(O)c1ccc2c(c1)C(C)(C)CC(C)(C)CC2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.35
RXRA P19793 3/20 0.35
RXRB P28702 1/20 0.35
RARA P10276 4/20 0.32
RARB P10826 4/20 0.32
RARG P13631 4/20 0.32
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
NOX1 Q9Y5S8 1/20 0.31
CSF1R P07333 1/20 0.30
CYP26A1 O43174 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP26B1 Q9NR63 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31085264 0.87 RXRA (0.41) UGT2B7RXRARXRBRARARARB
SCHEMBL8732926 0.81 RXRA (0.40) UGT2B7RXRARXRBRARARARB
SCHEMBL9419032 0.79 RXRA (0.38) UGT2B7RXRARXRBRARARARB
SCHEMBL11215262 0.76 RXRA (0.46) UGT2B7RXRARXRBRARARARB
SCHEMBL31003100 0.76 RXRA (0.40) UGT2B7RXRARXRBRARARARB
SCHEMBL9145102 0.74 NOX1 (0.36) UGT2B7MEN1TSHRKMT2ANOX1
SCHEMBL9770517 0.73 HPGD (0.41) RXRARXRBMEN1TSHRKMT2A
SCHEMBL3541162 0.73 RXRA (0.58) UGT2B7RXRARXRBRARARARB
SCHEMBL9418988 0.72 HTR2A (0.33) UGT2B7RXRARXRB
SCHEMBL9418950 0.70 RXRA (0.51) UGT2B7RXRARXRBRARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed
EP-0315071-A2 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed