SCHEMBL9423191

SCHEMBL9423191

NC(=O)n1nc(-c2ccco2)cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 7/20 0.56
PTGS2 P35354 1/20 0.48
HSD17B10 Q99714 4/20 0.46
CYP1A2 P05177 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 7/20 0.44
KDM4E B2RXH2 5/20 0.44
MEN1 O00255 4/20 0.44
RECQL P46063 4/20 0.44
CTDSP1 Q9GZU7 3/20 0.44
POLB P06746 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
MCL1 Q07820 2/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44
MAPT P10636 6/20 0.44
ALDH1A1 P00352 3/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9123670 0.84 PTGS1 (0.54) PTGS1PTGS2HSD17B10CYP1A2MAPK1
SCHEMBL3393181 0.73 KDM4E (0.53) PTGS1PTGS2HSD17B10CYP1A2MAPK1
SCHEMBL25407314 0.71 PTGS1 (0.56) PTGS1PTGS2HSD17B10KMT2AKDM4E
SCHEMBL25407369 0.70 PTGS1 (0.55) PTGS1PTGS2HSD17B10KDM4EMAPT
SCHEMBL9423332 0.69 LMNA (0.49) HSD17B10CYP1A2MAPK1CYP2C19KMT2A
SCHEMBL20488661 0.68 TDP1 (0.57) PTGS1HSD17B10KMT2AKDM4EMEN1
SCHEMBL2212356 0.68 PTGS1 (0.76) PTGS1PTGS2HSD17B10CYP1A2CYP2C19
SCHEMBL13425981 0.67 PTGS2 (0.46) PTGS1PTGS2HSD17B10CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL3169074 0.67 PTGS1 (0.74) PTGS1PTGS2HSD17B10CYP1A2CYP2C19
SCHEMBL930406 0.67 ADORA2A (0.63) ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5358947-A Treating hypertension, congestive heart failure AMERICAN CYANAMID COMPANY (US) 1994-10-25 US disclosed