SCHEMBL9424401

SCHEMBL9424401

CCc1sc(S(=O)(=O)NC(=O)Nc2ccc(Cl)cc2)cc1C.[NaH]

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 8/20 0.53
IDH1 O75874 5/20 0.48
KCNJ6 P48051 1/20 0.46
KCNJ5 P48544 1/20 0.46
KCNJ3 P48549 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KLKB1 P03952 1/20 0.45
CTSB P07858 1/20 0.45
ELANE P08246 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
MCL1 Q07820 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9424316 0.87 FBP1 (0.52) FBP1MEN1KMT2ALMNAMAPT
SCHEMBL9424273 0.84 IDH1 (0.49) IDH1KCNJ6KCNJ5KCNJ3ALDH1A1
SCHEMBL9424464 0.80 KMT2A (0.47) FBP1IDH1MEN1KMT2AKLKB1
SCHEMBL9424478 0.78 KMT2A (0.48) FBP1IDH1MEN1KMT2AKLKB1
SCHEMBL9424731 0.76 ALDH1A1 (0.51) IDH1MEN1KMT2AMAPTHTT
SCHEMBL9424704 0.75 ALDH1A1 (0.44) FBP1IDH1MEN1KMT2AKLKB1
SCHEMBL9424351 0.74 FBP1 (0.49) FBP1IDH1MEN1KMT2ALMNA
SCHEMBL9424721 0.73 MAPT (0.58) FBP1MEN1KMT2ALMNAMAPT
SCHEMBL8762900 0.73 CA12 (0.57) FBP1IDH1KCNJ6KCNJ5KCNJ3
SCHEMBL9424517 0.73 KMT2A (0.47) FBP1MEN1KMT2AKLKB1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5302724-A Thiophenesulfonylureas; anticarcinogenic agents ELI LILLY AND COMPANY (US) 1994-04-12 US disclosed
CN-1058401-A Anti-tumor compositions and methods of treatment LILLY CO ELI (US) 1992-02-05 CN disclosed
EP-0467613-A1 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1992-01-22 EP disclosed