SCHEMBL9428772

SCHEMBL9428772

CC(=O)c1ccc(OCCN2CCN(c3cc(=O)n(C)c(=O)n3C)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
ALDH1A1 P00352 1/20 0.56
HRH3 Q9Y5N1 10/20 0.56
RAB9A P51151 1/20 0.52
HRH1 P35367 3/20 0.51
HRH2 P25021 2/20 0.51
DRD3 P35462 2/20 0.49
DRD2 P14416 1/20 0.49
PSMB1 P20618 1/20 0.48
PSMB5 P28074 1/20 0.48
PSMB2 P49721 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428669 0.94 HRH3 (0.64) KDM4EHRH3HRH1HRH2DRD2
SCHEMBL9429182 0.93 HRH3 (0.64) KDM4EHRH3HRH1HRH2
SCHEMBL9429612 0.84 MEN1 (0.55) KDM4EALDH1A1RAB9ADRD3DRD2
SCHEMBL9429366 0.84 ALDH1A1 (0.52) KDM4EALDH1A1HRH1DRD3DRD2
Hydrochloric Acid SCHEMBL9428814 0.83 SIGMAR1 (0.54) KDM4EALDH1A1RAB9ADRD3DRD2
Hydrochloric Acid SCHEMBL9428580 0.83 MEN1 (0.51) ALDH1A1HRH1DRD3DRD2
SCHEMBL9429765 0.82 HRH3 (0.52) HRH3HRH1DRD2
SCHEMBL9428656 0.82 ALDH1A1 (0.50) ALDH1A1HRH3HRH1
SCHEMBL9429465 0.81 MAPT (0.52) KDM4EALDH1A1RAB9AHRH1DRD3
SCHEMBL9428719 0.81 HRH3 (0.47) KDM4EALDH1A1HRH3HRH1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed