SCHEMBL9428924

SCHEMBL9428924

CC=CC(=O)N(c1ccc(O)cc1)C1CCNC1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 17/20 0.44
SLC6A2 P23975 16/20 0.44
SLC6A3 Q01959 9/20 0.44
KCNH2 Q12809 5/20 0.41
CYP2D6 P10635 1/20 0.40
TRPM8 Q7Z2W7 2/20 0.39
NPY2R P49146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9429947 0.88 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9429217 0.86 SLC6A4 (0.47) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9429122 0.86 TRPM8 (0.51) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL8377826 0.84 SLC6A3 (0.40) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL8379418 0.82 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9428421 0.82 RAB9A (0.39) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9429926 0.82 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9842835 0.80 SLC6A2 (0.43) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL9428898 0.79 SLC6A4 (0.41) SLC6A4SLC6A2SLC6A3KCNH2TRPM8
SCHEMBL31142581 0.72 CHEK2 (0.42) SLC6A4SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5328907-A Treatment of allograft rejection in mammals and antiinflammatory agents SYNTEX (U.S.A.) INC. (US) 1994-07-12 US disclosed
US-5108999-A For treating inflammation, autoimmune disease or allograft rejection in mammals SYNTEX (U.S.A.) INC. (US) 1992-04-28 US disclosed
US-5001124-A 4-isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-03-19 US disclosed