SCHEMBL9429989

SCHEMBL9429989

O=c1cc(N2CCN(CCCOc3ccc(Cl)cc3)CC2)[nH]c(=O)[nH]1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.60
DRD2 P14416 7/20 0.54
HTR1A P08908 3/20 0.54
HTR2A P28223 3/20 0.54
DRD3 P35462 3/20 0.54
DRD1 P21728 1/20 0.54
DRD5 P21918 1/20 0.54
SIGMAR1 Q99720 4/20 0.53
TMEM97 Q5BJF2 2/20 0.53
HRH3 Q9Y5N1 8/20 0.51
HRH1 P35367 3/20 0.51
HRH2 P25021 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9428431 0.99 GPR84 (0.58) GPR84DRD2HTR1AHTR2ADRD3
SCHEMBL9428435 0.88 DRD2 (0.58) GPR84DRD2HTR1AHTR2ADRD3
Hydrochloric Acid SCHEMBL9428939 0.87 DRD2 (0.56) GPR84DRD2HTR1AHTR2ADRD3
SCHEMBL9429332 0.83 DRD2 (0.53) DRD2HTR1AHTR2ADRD3DRD1
SCHEMBL9428990 0.82 CYP1A2 (0.52) GPR84DRD2DRD3DRD1
SCHEMBL9428894 0.81 DRD2 (0.53) DRD2HTR1AHTR2ADRD3DRD1
SCHEMBL9429042 0.80 HTR2A (0.42) GPR84DRD2HTR2ADRD3DRD1
SCHEMBL9428251 0.78 DRD2 (0.48) DRD2HTR1AHTR2ADRD3DRD1
Oxalic Acid SCHEMBL9429238 0.76 MEN1 (0.55) DRD2HTR1AHTR2ADRD3SIGMAR1
SCHEMBL9429324 0.74 DRD2 (0.56) DRD2HTR1AHTR2ADRD3DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed