SCHEMBL9432011

SCHEMBL9432011

CCC(C)(C(=O)O)c1ccc(NN)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KIF11 P52732 1/20 0.37
NR1H4 Q96RI1 3/20 0.36
EPHX2 P34913 1/20 0.36
HDAC1 Q13547 1/20 0.35
NR3C2 P08235 1/20 0.35
TDP1 Q9NUW8 3/20 0.34
LMNA P02545 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
IDO1 P14902 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34
MAPT P10636 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9424924 0.81 MAPT (0.51) CYP1A2MEN1KMT2AHDAC1TDP1
SCHEMBL9433003 0.81 HDAC1 (0.46) CYP1A2MEN1KMT2AKIF11NR1H4
SCHEMBL9501933 0.80 MAPT (0.44) CYP1A2MEN1KMT2AEPHX2LMNA
SCHEMBL8494650 0.80 SMN1; SMN2 (0.47) CYP1A2MEN1KMT2ANR1H4EPHX2
SCHEMBL8148677 0.78 ESR1 (0.52) CYP1A2MEN1KMT2ALMNACYP3A4
SCHEMBL28915433 0.78 NPC1 (0.46) CYP1A2MEN1KMT2AKIF11LMNA
SCHEMBL1492728 0.77 CYP2C19 (0.50) CYP1A2KMT2AKIF11HDAC1CYP2D6
SCHEMBL15827159 0.77 CYP26B1 (0.40) CYP1A2MEN1KMT2AHDAC1CYP3A4
SCHEMBL20556837 0.77 MIF (0.48) CYP1A2MEN1KMT2ATDP1CYP3A4
SCHEMBL5794046 0.77 KDM4E (0.44) CYP1A2MEN1KMT2AKIF11HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5317103-A Migraine treatment MERCK SHARP & DOHME LIMITED (GB) 1994-05-31 US disclosed