SCHEMBL9435302

SCHEMBL9435302

N#C[C@]1(c2ccccc2)CC[C@H](N2CCN(CC(O)COc3ccc([N+](=O)[O-])cc3)CC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.58
TDP1 Q9NUW8 1/20 0.57
LMNA P02545 1/20 0.54
ALDH1A1 P00352 1/20 0.51
MAPT P10636 1/20 0.51
HTT P42858 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
RRM1 P23921 1/20 0.45
NPC1 O15118 1/20 0.43
CHRNA7 P36544 1/20 0.43
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435307 1.00 DRD4 (0.58) DRD4TDP1LMNAALDH1A1MAPT
SCHEMBL9435486 0.90 L3MBTL1 (0.56) DRD4L3MBTL1MEN1KMT2ARRM1
SCHEMBL9435493 0.90 L3MBTL1 (0.56) DRD4L3MBTL1MEN1KMT2ARRM1
SCHEMBL9098357 0.88 TSHR (0.52) MAPTL3MBTL1MEN1KMT2ARRM1
SCHEMBL9098349 0.88 TSHR (0.52) MAPTL3MBTL1MEN1KMT2ARRM1
SCHEMBL9098366 0.88 TSHR (0.52) MAPTL3MBTL1MEN1KMT2ARRM1
SCHEMBL9435669 0.86 MAPT (0.59) MAPT
SCHEMBL9435672 0.86 MAPT (0.59) MAPT
SCHEMBL9435568 0.83 TSHR (0.54) MAPTHTTMEN1KMT2ARRM1
SCHEMBL9435578 0.83 TSHR (0.54) MAPTHTTMEN1KMT2ARRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371088-A 1-aryl-4-piperazinylcyclohexanecarbonitriles, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed