SCHEMBL9435641

SCHEMBL9435641

N#C[C@]1(c2ccccc2)CC[C@H](N2CCN(CC(O)CSc3ccccc3)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.44
CYP2D6 P10635 1/20 0.41
KDM1A O60341 1/20 0.41
OPRM1 P35372 2/20 0.40
OPRD1 P41143 1/20 0.40
OPRL1 P41146 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRM4 P08173 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435647 1.00 MAPT (0.44) MAPTCYP2D6KDM1AOPRM1OPRD1
Benzene SCHEMBL9435651 0.85 CYP2D6 (0.44) CYP2D6KDM1AOPRM1OPRD1OPRL1
SCHEMBL9435749 0.84 OPRM1 (0.48) CYP2D6KDM1AOPRM1OPRD1ADRA1D
SCHEMBL9435756 0.84 OPRM1 (0.48) CYP2D6KDM1AOPRM1OPRD1ADRA1D
SCHEMBL9435486 0.82 L3MBTL1 (0.56) CYP2D6MEN1KMT2A
SCHEMBL9435493 0.82 L3MBTL1 (0.56) CYP2D6MEN1KMT2A
SCHEMBL9435662 0.78 CYP2D6 (0.44) CYP2D6KDM1AOPRM1OPRD1CA12
SCHEMBL9435657 0.78 CYP2D6 (0.44) CYP2D6KDM1AOPRM1OPRD1CA12
SCHEMBL9098349 0.78 TSHR (0.52) MAPTCYP2D6MEN1KMT2A
SCHEMBL9435760 0.78 HTR1A (0.48) MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371088-A 1-aryl-4-piperazinylcyclohexanecarbonitriles, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed