SCHEMBL9436714

SCHEMBL9436714

Cn1c(N(CCO)CCNCCCCc2ccc(Cl)cc2)cc(=O)n(C)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 1/20 0.43
ADRB1 P08588 1/20 0.43
SLC6A4 P31645 1/20 0.43
KCNH2 Q12809 1/20 0.43
SLC47A2 Q86VL8 1/20 0.43
SLC47A1 Q96FL8 1/20 0.43
RXFP1 Q9HBX9 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
TP53 P04637 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
P2RX3 P56373 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
ADRB2 P07550 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428345 0.94 SLC22A2 (0.40) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9385340 0.86 KCNH2 (0.60) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9428759 0.86 ADRB2 (0.38) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9429025 0.84 ADRB1 (0.36) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9389045 0.83 KCNH2 (0.61) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9429655 0.81 ADRB2 (0.39) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9428363 0.81 KCNH2 (0.40) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9388183 0.80 KCNH2 (0.57) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9869584 0.76 KCNH2 (0.52) SLC22A2ADRB1SLC6A4KCNH2SLC47A2
SCHEMBL9388214 0.75 TAAR1 (0.48) SLC22A2ADRB1SLC6A4KCNH2SLC47A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed